出版年 | 標題 | 作者 | 系所 |
2011 | 1,1-二氧化苯駢[1.3.2]二噻唑亞烷衍生物作為第二型環氧化酶
與第五型脂氧合酶雙效抑制劑之設計、合成與活性評估 Design, Synthesis and Biological Evaluation of
Benzo[1.3.2]dithiazolium Ylide 1,1-Dioxide Derivatives as
Dual Cyclooxygenase-2/5-Lipoxygenase Inhibitors | Chen-Ming Tan; 譚誠明 | 藥學研究所 |
2006 | Quinoline 衍生物之設計、合成與生物活性評估 Design,Synthesis and Biological Evaluation of Quinoline Analogues | RAHUL SUBHASH TALEKAR; 塔立卡 | 藥學研究所 |
2007 | Suberoylanilide Hydroxamic Acid (SAHA)類似物作為潛能抗癌藥物之設計與合成 Design and Synthesis of Suberoylanilide Hydroxamic Acid (SAHA) Homologues as Potential Antitumor Agents | Sheng-Ju Hsu; 徐聖如 | 藥學研究所 |
2018 | 兼具誘導神經元生長之膽鹼酯酶抑制劑作為阿茲海默症潛在治療藥物 The Neurite Outgrowth Inducer with Cholinesterase Inhibitory Activities as Potential Agent for Anti-Alzheimer's Disease | 馮湘芷; Sheang-Tze Fung | 藥學研究所 |
2012 | 喹唑啉酮類化合物作為組蛋白去乙醯脢抑制劑之設計
合成及其生物活性研究 Design, Synthesis, and Biological Evaluation of Quinazolinone Derivatives as Histone Deacetylase (HDAC) Inhibitors | Chao-Wu Yu; 余兆武 | 藥學研究所 |
2005 | 喹啉衍生物作為癌細胞毒殺劑之設計與合成 Design and Synthesis of Quinoline Derivatives as Potential Cytotoxic Agents | Yin-Ling Wei; 魏吟玲 | 藥學研究所 |
2018 | 新穎性第六亞型組蛋白去乙醯酶抑制劑在膠質母細胞瘤之抗癌作用機轉探討 Investigation of the anticancer mechanisms of a novel HDAC6 inhibitor in glioblastoma | 劉佳蓉; Jia-Rong Liu | 藥學研究所 |
2017 | 潛質抗癌藥物MTH1抑制劑之設計合成 與生物活性評估 Design, Synthesis and Biological Evaluation of MTH1 Inhibitors as Potential Anti-cancer Agents | 程澤華; Ze-Hua Cheng | 藥學研究所 |
2009 | 神經滋養調控劑之合成設計與生物活性評估 Design, Synthesis and Evaluation of Neurotrophic Modulators | Fei-Chiao Kuo; 郭斐荍 | 藥學研究所 |
2017 | 苯并咪唑衍生物作為間變性淋巴瘤激酶/組蛋白去乙醯酶雙重抑製劑之設計與合成 Design and Synthesis of Benzimidazole Derivatives as Anaplastic Lymphoma Kinase / Histone Deacetylase Dual Inhibitors | I-Chun Lin; 林怡君 | 藥學研究所 |
2013 | 設計合成具有多重功效之羥烷基取代八羥基/烷氧基喹啉衍生物作為治療阿茲海默症之活性評估 Design, Synthesis and Biological Evaluation of Hydroxyalkyl Substituted 8-Hydroxyl/Alkoxyquinolines with Multifunctional Activities against Alzheimer’s Disease | Chen-Wei Huang; 黃振瑋 | 藥學研究所 |
2014 | 設計合成與評估8-甲氧基喹啉衍生物作爲抗阿茲海默症之潛在多靶點藥物 Design, Synthesis and Evaluation of 8-Methoxyquinoline Derivatives as Potential Multifunctional Agents for the Treatment of Alzheimer’s Disease | Qing-Qing Ye; 葉青青 | 藥學研究所 |
2016 | "設計和合成2-胺基3,4-二氫喹唑啉衍生物作為潛在β位澱粉樣前體蛋白切割酵素抑制劑" Design and Synthesis of 2-Amino-3,4-dihydroquinazoline Derivative as Potential β-site amyloid precursor protein cleaving enzyme 1 (BACE 1)Inhibitors | Guan-Yun Chen; 陳冠勻 | 藥學研究所 |
2010 | 設計與合成1,4-二甲基咔唑及橢圓玫瑰樹鹼之
苯磺醯胺衍生物作為潛能抗癌試劑 Design and Synthesis of 1,4-Dimethylcarbazole and Ellipticine Analogues Containing Benzenesulfonamide Moiety as Potential Anti-cancer Agents | Hsueh-Yun Lee; 李學耘 | 藥學研究所 |
2012 | 設計與合成4-芳香基-1-苯甲基喹唑啉-2-酮類化合物作為第六亞型組蛋白去乙醯酶抑制劑之可行性 Design and Synthesis of 4-Aryl-1-benzylquinazolin-2-one Derivatives as Potential Histone Deacetylase 6 (HDAC6) Inhibitors | Fang-Yu Kan; 闞方妤 | 藥學研究所 |
2010 | 設計與合成4-芳香基-1-苯甲基喹唑啉酮衍生物作為第四型與第五型磷酸二酯酶雙效抑制劑 Design and Synthesis of 4-Aryl-1-benzyl-1H-quinazolin-2-ones
as Dual Phosphodiesterase 4 and 5 Inhibitors | Chih-Yi Chang; 張智億 | 藥學研究所 |
2013 | 設計與合成吲哚-2-酮衍生物作為潛能蛋白激酶 抑制劑及其活性評估 Design, Synthesis and Biological Evaluation of Indolin-2-one
Derivatives as Potential Kinase Inhibitors | Ajit Dhananjay Jagtap; 杰合南 | 藥學研究所 |
2012 | 設計與合成吲哚-2-酮衍生物作為潛能蛋白激酶抑制劑及其活性評估 Design, Synthesis and Biological Evaluation of Indolin-2-one Derivatives as Potential Protein Kinase Inhibitors | Hsiao-Chun Wang; 王筱君 | 藥學研究所 |
2012 | 設計與合成喹唑啉-2-酮衍生物作為潛能第五型磷酸二
酯酶抑制劑之可行性評估 Design, Synthesis and Feasibility Evaluation of 1H-Quinazolin-2-one Derivatives as Potential
PhosphodiesteraseⅤInhibitors | Chun-Wei Lo; 羅浚瑋 | 藥學研究所 |
2018 | 設計與合成喹唑啉和喹啉衍生物作為蛋白激酶抑制劑及生物活性評估 Design, Synthesis, and Biological Evaluation of Quinazoline and Quinoline Derivatives as Kinase Inhibitors | 吳昆達; Kuen-Da Wu | 藥學研究所 |